Transporter Symbol

Substrate

VACHT, SLC18A3

acetylcholine

ANT1, T1, PEO2, PEO3, SLC25A4

ADP

ANT2, SLC25A5, 2F1, T2, SLC25A5

ADP

SVCT2, KIAA0238, YSPL2, SLC23A1

ascorbic acid

BGT-1, SLC6A12

betaine, gama-aminobutyric acid

AE1, RTA1A, SLC4A1

bicarbonate, chloride

AE2, HKB3, SLC4A2

bicarbonate, chloride

AE3, bAE3, SLC4A3, SLC2C

bicarbonate, chloride

SMVT, SLC5A6

biotin, pantothenate, lipoate

Aralar, SLC25A12

Ca2+

Aralar-like, CTLN2, SLC25A13

Ca2+

NCKX1, KIAA0702, SLC24A1

Ca2+

NCX1, SLC8A1

Ca2+

OCTN1, SLC22A4

carnitine, organic cation

OCTN2, SCD, CDSP, SLC22A5

carnitine, organic cation

CTP, SLC25A1

citrate

CFTR

Cl-

CTR-1, hCTR1, COPT1, SLC31A1

copper

CTR-2, hCTR2, COPT2, SLC31A2

copper

CRTR, SLC6A8, CT1

creatine

CT-2, SLC6A10

creatine

rBAT, SLC3A1, D2, D2H, CSNU1, SLC3A1

cystine, dibasic and neutral amino acids

PEPT1, hPEPT1, SLC15A1

Di/tripeptides

4F2, 4F2HC, MDU1, NACAE, 4T2HC, SLC3A2

dibasic and neutral amino acids

DIC, SLC25A10

dicarboxylates

SDCT1, SLC13A2, NADC1, NADC-1

dicarboxylates

DAT

Dopamine

MRP1, ABCC1, MRP, GS-X

drug conjugates

MRP3, ABCC3, MLP2, ABC31, MOAT-D, CMOAT2, EST90757

drug conjugates

NRAMP1, LSH, SLC11A1

Fe2+

NRAMP2, DCT1, SLC11A2,

Fe2+, Mn2+, Zn2+

GAT-2, SLC6A13

gama-aminobutyric

GAT3, GAT-3, SLC6A11

gama-aminobutyric

GAT1, GAT-1, SLC6A1

gama-aminobutyric acid

GLUT1, SLC2A1, GLUT

glucose, dehydroascobic acid

GLUT3, SLC2A3

glucose, dehydroascorbic acid

GLUT4, SLC2A4

glucose, dehydroascorbic acid

GLUT2, SLC2A2

glucose, fructose

GLUT5, SLC2A5

glucose, fructose

BCMP1, UCP4, SLC25A14

H+

NHE1, SLC9A1, APNH

H+

NHE2, SLC9A2

H+

NHE3, SLC9A3/3P

H+

NHE4, SLC9A4

H+

NHE5, SLC9A5

H+

NHE6, KIAA0267, SLC9A6

H+

UCP1 , UCP

H+

UCP2, SLC25A8

H+

UCP3, SLC25A9

H+

NTCP2, ISBT, SLC10A2

ileal sodium-dependent

SMIT, SLC5A3

Inositol

NIS, SLC5A5

Iodide

KCC1, SLC12A4

K+/Cl-

KCC3, SLC12A6

K+/Cl-

KCC4, SLC12A7

K+/Cl-

SATT, SLC1A4, ASCT1

L-Ala, L-Ser, L-Cys

ATBo, SLC1A5, RDRC, hATBo, ASCT2, AAAT, M7V1, RDRC

L-Ala, L-Ser, L-Thr, L-Cys, L-Gln

CAT-4, SLC7A4, CAT4, HCAT3

L-Arg

LAT2, LAT-2, y+LAT-2, KIAA0245, SLC7A6

L-Arg

LAT3, LAT-3, LPI, y+LAT-1, SLC7A7

L-Arg

CAT1, HCAT1, ERR, REC1L, SLC7A1, ATRC1, CAT-1

L-Arg, L-Lys, L-Orn

CAT2, SLC7A2, CAT-2a, CAT-2b, ATRC2, HCAT2

L-Arg, L-Lys, L-Orn

EAAT1, SLC1A3, GLAST, GLAST1

L-Glu, D, L-Asp

EAAT2, SLC1A2, GLT-1

L-Glu, D, L-Asp

EAAT3, SLC1A1, EAAC1

L-Glu, D, L-Asp

EAAT4, SLC1A6

L-Glu, D, L-Asp

EAAT5, SLC1A7

L-Glu, D, L-Asp

GLYT1

L-Glycine

GLYT2, GLYT-2, NET1, SLC6A5

L-Glycine

FATP4, SLC27A4

long fatty acids

PROT, SLC6A7

L-Proline

ABCC4, MOAT-B, MRP4, EST170205

methotrexate

SVMT, SLC18A2, VMAT2

monoamine

VAT1, SLC18A1, VMAT1, CGAT

monoamine

MCT1, SLC16A1, MCT

monocarboxylic acids

MCT2, SLC16A7

monocarboxylic acids

MCT3, SLC16A3

monocarboxylic acids

MCT5, SLC16A5

monocarboxylic acids

MCT6, SLC16A6

monocarboxylic acids

MCT4, SLC16A4

monocarboxylic acidsmonocarboxylic acids

NCCT, SLC12A3, TSC, hTSC

Na+/K+/Cl-

NKCC1, SLC12A2

Na+/K+/Cl-

NKCC2, SLC12A1

Na+/K+/Cl-

SGLT1, SLC5A1, D22S675

Na+-glucose

SGLT2, SLC5A2

Na+-glucose

DTD, SLC26A2

Na+-sulfate

GLUT6, SLC2A3P, GLUT3P1

No (pseudogene)

NAT1, SLC6A2, NET1, SLC6A5

Norepinephrine

CNT1, SLC28A1, cit, N2, SLC28A1, HCNT1

nucleosides

CNT2, SLC28A2, cif, N1, SPNT1, HCNT2

nucleosides

ENT1(es), SLC29A1, hENT1

nucleosides

ENT2(ei), HNP36, SLC29A2, DER12

nucleosides

LST-1, SLC21A6, OATP-C

organic anions

OAT1, PAHT, ROAT1, SLC22A6

organic anions

OAT2, OAT-2, NLT, SLC22A7

organic anions

OAT3, SLC22A8

organic anions

OAT4

organic anions

OAT-K1, OAT-K2, SLC21A4

organic anions

OATP, OATP1, SLC21A3

organic anions

OATP2, SLC21A5

organic anions

OATP3, SLC21A7

organic anions

OATP5, SLC21A13

organic anions

OATP8, SLC21A8

organic anions

OCT1, SLC22A1, hOCT1

organic cations

OCT2, SLC22A2, NLT, hOCT2

organic cations

ORNT1, D13S327, HHH, SLC25A15

ornithine

TAP1

peptides

TAP2, ABCB3, D6S217E, PSF2, RING11

peptides

GLVR1, PiT-1, SLC20A1

phosphate

NAPI-3B, SLC34A2

phosphate

NPT1, SLC17A1, NAPI-1

phosphate

NPT2, SLC34A1, NAPI-3, SLC17A2

phosphate

PGT, SLC21A2

prostaglandins

SPNT1a, hSPNT1a

purine nucleosides

MCT7, SLC16A2, XPCT, DXS128

putative transporter

FOLT, SLC19A1, RFC1, REFC, CHMD

reduced folates

HTT, SERT, SLC6A4

serotonin

NBC1, NBC2, pNBC, HNBC1, hhNMC, SLC4A4

sodium, bicarbonate

Transporter Isoform Symbol

Substrate/Drug

SUR1, ABCC8, HI, PHHI, SUR, MRP8, HRINS

sulfonylureas

SUR2

sulfonylureas

TAUT, SLC6A6

taurine

NTCP, NTCP1, SLC10A1

taurocholate

ABCP, BCRP, ABCG2, MXR, ABC15, EST157481

Tc-Tetrofosmin (radiopharmaceutical substrate)

MDR1, ABCB1, PGY1, P-gp

various

MDR2, MDR3, ABCB4, PGY3, PFIC-3

various

ZNT1, ZNT-1, SLC30A1

zinc

ZNT2, SLC30A2

zinc

ZNT3, ZNT-3, SLC30A3

zinc

ZNT4, ZNT-4, SLC30A4

zinc